BDBM503565 US11034670, Ex. 5

SMILES Clc1cc(ccc1N1CCN(CC1)C(=O)CCc1nc(=O)c2ccccc2[nH]1)C(=O)NC1CCC1

InChI Key InChIKey=VKZNGDOKTNBOCZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 503565   

TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Mitobridge

US Patent
LigandPNGBDBM503565(US11034670, Ex. 5)
Affinity DataIC50:  51nMAssay Description:The scintillation proximity assay (SPA) is designed to measure PARP activity using purified recombinant PARP-1 enzyme and is ideal for high throughpu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent