BDBM50359260 CHEMBL1923611

SMILES CCC[C@@H]1NCCOc2ccccc2CCCNC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)N(C)C1=O

InChI Key InChIKey=HVNSCQHWQRWMCW-IEZKXTBUSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50359260   

TargetAppetite-regulating hormone(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359260(CHEMBL1923611)
Affinity DataKi:  16nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAppetite-regulating hormone(Homo sapiens (Human))
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359260(CHEMBL1923611)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed