BDBM50369893 CHEMBL1201959

SMILES C1CCC(CC1)C1NC(Cc2c1[nH]c1ccccc21)c1nc(c[nH]1)-c1ccccc1

InChI Key InChIKey=CMKNFFUUKQPJOF-UHFFFAOYSA-N

Data  5 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50369893   

TargetSomatostatin receptor type 3(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50369893(CHEMBL1201959)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [125 I -Tyr]SRIF-14 binding to membranes isolated from CHO-K1 cells expressing cloned human SRIF receptor (sst-3) subtypeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50369893(CHEMBL1201959)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of [125 I -Tyr]SRIF-14 binding to membranes isolated from CHO-K1 cells expressing cloned human SRIF receptor (sst-1) subtypeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50369893(CHEMBL1201959)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125 I -Tyr]SRIF-14 binding to membranes isolated from CHO-K1 cells expressing cloned human SRIF receptor (sst-4) subtypeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50369893(CHEMBL1201959)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125 I -Tyr]SRIF-14 binding to membranes isolated from CHO-K1 cells expressing cloned human SRIF receptor (sst-2) subtypeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50369893(CHEMBL1201959)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125 I -Tyr]SRIF-14 binding to membranes isolated from CHO-K1 cells expressing cloned human SRIF receptor (sst-5) subtypeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50369893(CHEMBL1201959)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration required to inhibit SRIF-14 induced reduction of cAMP in CHO-K1 cells expressing the human sst3 receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed