BDBM50380922 CHEMBL2016739

SMILES CN([C@H]1CC[C@]2(CC1)OC(=O)c1ccncc21)C(=O)Nc1cnc(cn1)-c1ccccc1

InChI Key InChIKey=PZHDBZKHTKEPPX-SMQSCJQKSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50380922   

TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380922(CHEMBL2016739)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]PPY from human recombinant NPYY5 receptor expressed in insect Sf9 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380922(CHEMBL2016739)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human NPYY1 assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed