BDBM50393024 CHEMBL2152689::US9656959, Example 54
SMILES OC[C@H](NC(=O)c1ccccn1)C(=O)Nc1cccc(n1)-c1ccc(Oc2ccc(F)cc2)cc1
InChI Key InChIKey=WVFJNTNBBZOWRT-QHCPKHFHSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50393024
Affinity DataKi: 195nMAssay Description:Blockade of Nav1.7 by electrophysiological patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:In vitro assays were performed in a recombinant cell line expressing cDNA encoding the alpha subunit (Nav1.7, SCN9a, PN1, NE) of human Nav1.7 (Access...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Blockade of Nav1.7 by FLIPR TETRA sodium dye assay in presence of KCl saltMore data for this Ligand-Target Pair