BDBM50395012 CHEMBL2163456::US9708370, 58 CP-3(ii)
SMILES C[C@H](NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](N)Cc1cnc[nH]1)C(=O)NN(Cc1ccccc1)C(=O)N[C@H](C)C(=O)N[C@@H](CCCCN)C(N)=O
InChI Key InChIKey=WYDHGNGESNONNQ-KDSGNBONSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50395012
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
TargetEstrogen receptor [D538G](Homo sapiens (Human))
Valorisation-Recherche, Limited Partnership
US Patent
Valorisation-Recherche, Limited Partnership
US Patent
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair