BDBM50396827 CHEMBL1712297

SMILES ONC(=O)CN1C(=O)C2(OCCO2)c2cc(Br)ccc12

InChI Key InChIKey=DDNUPCQCTVYXNK-UHFFFAOYSA-N

Data  1 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50396827   

TargetAminopeptidase N(Sus scrofa (Pig))
Shandong Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50396827(CHEMBL1712297)
Affinity DataKi:  2.79E+3nMAssay Description:Inhibition of porcine kidney microsome aminopeptidase using L-Leu-p-nitroanilide as substrate by Dixon methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50396827(CHEMBL1712297)
Affinity DataIC50:  360nMAssay Description:Inhibition of pig kidney microsome aminopeptidase-N using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50396827(CHEMBL1712297)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of aminopeptidase-N in human ES2 cells using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Shandong Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50396827(CHEMBL1712297)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of porcine kidney microsome aminopeptidase using L-Leu-p-nitroanilide as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed