BDBM50399572 CHEMBL2180931
SMILES C[C@H](Nc1nc2nn(C)cc2c2nc(nn12)-c1ccco1)c1ccccc1
InChI Key InChIKey=OWWOFJVMVLDYOC-LBPRGKRZSA-N
Data 8 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50399572
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 55.2nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 338nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 338nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.29E+3nMAssay Description:Antagonist activity at human A2B receptor expressed in CHO cell membrane assessed as reduction in NECA-stimulated adenylyl cyclase activity in presen...More data for this Ligand-Target Pair
Affinity DataKi: 5.29E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as NECA-induced adenylate cyclase activityMore data for this Ligand-Target Pair