BDBM50405117 CHEMBL4170869

SMILES COc1ccc(cc1)N1C(=O)\C(=C/c2ccccc2)C1(C(=O)NC1CCCCC1)c1cc(F)c(F)c(F)c1

InChI Key InChIKey=IFNIJFNEVBNCCA-WADGIJBFSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50405117   

TargetHistamine H3 receptor(Homo sapiens (Human))
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405117(CHEMBL4170869)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human H3R expressed in HEK293 cells harboring glosensor-22F cAMP plasmid DNA assessed as inhibition of forskolin-stimulated cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Csir-Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50405117(CHEMBL4170869)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human H3R expressed in HEK293 cells harboring glosensor-22F cAMP plasmid DNA assessed as inhibition of forskolin-stimulated cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed