BDBM50419878 CHEMBL1956195
SMILES CC(Oc1ccccc1CC1CC1)C1=NCCN1
InChI Key InChIKey=SEKAQUSPSDPIAN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 18 hits for monomerid = 50419878
Affinity DataKi: 10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Binding affinity at human alpha2B ARMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2B expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human alpha2C adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells after 240 secs by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.31E+3nMAssay Description:Agonist activity at human alpha2B adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
Affinity DataEC50: 3.31E+3nMAssay Description:Agonist activity at human alpha2B ARMore data for this Ligand-Target Pair
Affinity DataEC50: 3.31E+3nMAssay Description:Agonist activity at human adrenoceptor aplha 2B expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair