BDBM50428826 CHEMBL2337127

SMILES [#6]-[#8]-c1cc(-[#6]-[#6]-c2ccccc2)c(-[#6](-[#8])=O)c(-[#8])c1-[#6]\[#6]=[#6](/[#6])-[#6]-[#6]\[#6]=[#6](\[#6])-[#6]

InChI Key InChIKey=DKNIJLWIVUCTHW-CPNJWEJPSA-N

Data  3 Kd  2 EC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50428826   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Max Planck Institute For Molecular Genetics

Curated by ChEMBL
LigandPNGBDBM50428826(CHEMBL2337127)
Affinity DataEC50:  73nMAssay Description:Agonist at human PPARgamma LBD expressed in human HEK293 cells cotransfected with GAL4-Luc assessed as transcriptional activation by luciferase repor...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Max Planck Institute For Molecular Genetics

Curated by ChEMBL
LigandPNGBDBM50428826(CHEMBL2337127)
Affinity DataKd:  19nMAssay Description:Binding affinity to human PPARgamma (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Max Planck Institute For Molecular Genetics

Curated by ChEMBL
LigandPNGBDBM50428826(CHEMBL2337127)
Affinity DataEC50:  50nMAssay Description:Agonist at human PPARgamma LBD expressed in human HEK293 cells cotransfected with GAL4-Luc assessed as transcriptional activation by luciferase repor...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Helmholtz Centre For Infection Research

Curated by ChEMBL
LigandPNGBDBM50428826(CHEMBL2337127)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to human PPARalpha (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre For Infection Research

Curated by ChEMBL
LigandPNGBDBM50428826(CHEMBL2337127)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to human PPARdelta (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed