BDBM50436201 FLUTRIMAZOLE::UR-4056
SMILES Fc1ccc(cc1)C(c1ccccc1)(c1ccccc1F)n1ccnc1
InChI Key InChIKey=QHMWCHQXCUNUAK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50436201
Affinity DataIC50: 1.38E+4nMAssay Description:Antagonist activity at human GTS-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
City Of Hope National Medical Center
Curated by ChEMBL
City Of Hope National Medical Center
Curated by ChEMBL
Affinity DataEC50: 6.10E+3nMAssay Description:Agonist activity at PXR (unknown origin) expressed in human HepG2 cells assessed as induction of CYP3A4 transactivation after 16 hrs by luciferase re...More data for this Ligand-Target Pair