BDBM50440111 CHEMBL2426127

SMILES CC(C)(CNC(=O)Cc1ccccc1)[C@@H](c1ccccc1)c1ccc2n(ncc2c1)-c1ccc(F)cc1

InChI Key InChIKey=IKUATMHYCWRCHC-HKBQPEDESA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50440111   

TargetGlucocorticoid receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50440111(CHEMBL2426127)
Affinity DataEC50:  2.52E+3nMAssay Description:Transrepression activity at glucocorticoid receptor in human A549 cells assessed as inhibition of PMA-stimulated AP1 response element by luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50440111(CHEMBL2426127)
Affinity DataEC50:  977nMAssay Description:Transactivation activity at glucocorticoid receptor ligand binding domain (unknown origin) expressed in human Hela cells co-expressing GAL4 DNA bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed