BDBM50442686 CHEMBL2442300

SMILES CN(C)CCNc1ccn2ncc(-c3ccc4ccccc4c3)c2n1

InChI Key InChIKey=AVLJGDZDWUWISV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442686   

TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50442686(CHEMBL2442300)
Affinity DataIC50:  5nMAssay Description:Inhibition of Pim1 (unknown origin) using STK3 as substrate preincubated for 30 mins followed by substrate and ATP addition after 45 mins by HTRF ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed