BDBM50445227 CHEMBL3102955
SMILES Oc1ccc(cc1O)-c1c[nH]c2ncc(cc12)-c1ccc(O)c(O)c1
InChI Key InChIKey=CJTAMMDFIMBFDQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50445227
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Competitive inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using ATP as subst...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein c...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein c...More data for this Ligand-Target Pair