BDBM50446891 CHEMBL3115314::US10246442, Example 61::US10975062, Example 61
SMILES OC(=O)c1cnn(c1)-c1nc(N2CCCC2)c2cc(Oc3ccc(Cl)cc3)ccc2n1
InChI Key InChIKey=YEHGRYMGRBBRMA-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50446891
Affinity DataIC50: 50nMAssay Description:Inhibition of PHD2 (181 to 417) (unknown origin) using HIF-1alpha peptide as substrate assessed as 2-Oxoglutarate conversion to succinic acid preincu...More data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:The PHD enzymatic assay was performed in 0.5 ml of reaction mixture containing the following: purified PHD2181-417 polypeptide (3 μg), synthetic...More data for this Ligand-Target Pair