BDBM50450512 CHEMBL4172787

SMILES O[C@H]1CN(C[C@@H]1Oc1ccc(C#N)c(F)c1)S(=O)(=O)c1ccc(Cl)cc1Cl

InChI Key InChIKey=WXXLTRAHCCRGDR-HOTGVXAUSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50450512   

TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
TBA

Curated by ChEMBL

LigandBDBM50450512(CHEMBL4172787)Copy SMILESCopy InChI

Affinity DataIC50:  40nMAssay Description:Antagonist activity at human TRPV4 expressed in BHK/AC9 or HEK MSR2 cells assessed as inhibition of PF-04674114-induced Ca2+ flux pre-incubated for 1...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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