BDBM50451040 CHEMBL4218771

SMILES Cl.Fc1ccc(cc1)C(N1CCN(CCNC(=O)c2ccccn2)CC1)c1ccc(F)cc1

InChI Key InChIKey=OKODSFKDPWCAAS-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50451040   

Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451040(CHEMBL4218771)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]mesulergine from serotonin 5-HT2C receptor in Sprague-Dawley rat brain cortex homogenates incubated for 15 mins by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451040(CHEMBL4218771)
Affinity DataKi:  218nMAssay Description:Displacement of [3H]ketanserin from serotonin 5-HT2A receptor in Sprague-Dawley rat brain cortex homogenates incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451040(CHEMBL4218771)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from serotonin 5-HT1A receptor in Sprague-Dawley rat brain cortex homogenates incubated for 30 mins by liquid scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed