BDBM50461709 CHEMBL4225349
SMILES Clc1ccc(cc1)-n1c(nc2c(ncnc12)N1CCN(Cc2ccccc2Cl)CC1)-c1ccccc1Cl
InChI Key InChIKey=SXOSAVAARDEMIU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50461709
Affinity DataKi: 8nMAssay Description:Displacement of [3H]CP55940 from human CB1 expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Rti International
Curated by ChEMBL
Rti International
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]astemizole from human ERG expressed in HEK cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 462nMAssay Description:Inverse agonist activity human CB1 expressed in CHOK1 cells co-expressing Galpha-q16 incubated for 60 secs by Calcein-4 AM dye-based FLIPR assayMore data for this Ligand-Target Pair