BDBM50466254 CHEMBL4288569
SMILES CN(C)CCN1CCN(CC1)c1nc(NCc2cccc(Cl)c2)c2cc(ccc2n1)-c1ccc(=O)n(C)c1
InChI Key InChIKey=POKZINYHLOHGEB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50466254
TargetBromodomain-containing protein 2(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 27nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD2 isoform 1 bromodomain 1/2 (K71 to D455 residues) expressed...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD3 bromodomain 1/2 (P24 to P416 residues) expressed in Escher...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 21nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD3 bromodomain 2 (G306 to P416 residues) expressed in Escheri...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 18nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD4 long isoform bromodomain 1 (N44 to E168 residues) expresse...More data for this Ligand-Target Pair
3D Structure (crystal)TargetBromodomain testis-specific protein(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 67nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRDT isoform b bromodomain 1/2 (N21 to E382 residues) expressed...More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 20nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRDT isoform b bromodomain 1 (N21 to E137 residues) expressed i...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 44nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD4 long isoform bromodomain 1/2 (N44 to E460 residues) expres...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 50nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD4 long isoform bromodomain 2 (K333 to E460 residues) express...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 21nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD3 bromodomain 1 (P24 to E144 residues) expressed in Escheric...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 33nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD2 isoform 1 bromodomain 1 (K71 to N194 residues) expressed i...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 24nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRD2 isoform 1 bromodomain 2 (E348 to D455 residues) expressed ...More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKd: 160nMAssay Description:Displacement of biotinylated acetylated peptide from recombinant human partial length BRDT isoform b bromodomain 2 (K250 to E382 residues) expressed ...More data for this Ligand-Target Pair