BDBM50468502 CHEMBL4289527
SMILES CCN(CC)c1cc2n(C)c(=O)c(=O)n(C)c2cc1NC(=O)c1ccccc1OC
InChI Key InChIKey=ATFDQVXQRDPKSI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50468502
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataKd: 9.70E+3nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair