BDBM50468514 CHEMBL4277790
SMILES CCOc1ccccc1C(=O)Nc1cc2n(C)c(=O)c(=O)n(C)c2cc1N1CCC(C)CC1
InChI Key InChIKey=DKHUINVTTPXRJP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50468514
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair