BDBM50493178 CHEMBL2419581
SMILES C(Cc1c[nH]c2ccccc12)Nc1ccc(CN2CCOCC2)cc1
InChI Key InChIKey=UCTRCZYTETZMOI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50493178
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]-(R)-alpha-methylhistamine from human histamine H3 receptor expressed in HEK293 cells after 90 to 120 mins by liquid scintillatio...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells assessed by forskolin induced cAMP response element activation after 5 h...More data for this Ligand-Target Pair