BDBM50500206 CHEMBL3746828

SMILES FC1COc2ccc(cc2OC1)S(=O)(=O)N[C@@H](c1cc2ccccc2s1)c1ccccc1Cl

InChI Key InChIKey=JRUJLWQVCJSIOM-OODIQHKMSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50500206   

TargetGlucokinase regulatory protein(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50500206(CHEMBL3746828)
Affinity DataEC50:  4.10E+3nMAssay Description:Inhibition of glucokinase-GKRP binding interaction in mouse hepatocytes assessed as induction of glucokinase translocationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucokinase regulatory protein(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50500206(CHEMBL3746828)
Affinity DataIC50:  74nMAssay Description:Binding affinity to human biotinylated AviTag GKRP assessed as inhibition of protein interaction with fluorescein tagged human glucokinase by AlphaSc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed