BDBM50517754 CHEMBL4456660

SMILES CC(C)C[C@H](NC(=O)NCc1cn(nn1)-c1ccccc1COC(=O)c1cccc2ccccc12)C(=O)NO

InChI Key InChIKey=AARBAVOFBGGQFJ-DEOSSOPVSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50517754   

TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50517754(CHEMBL4456660)
Affinity DataIC50:  32nMAssay Description:Inhibition of porcine kidney microsomal APN using L-Leu-p-nitroanilide as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50517754(CHEMBL4456660)
Affinity DataIC50:  810nMAssay Description:Inhibition of APN on human PLC/PRF/5 cell surface using L-Leu-p-nitroanilide as substrate after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50517754(CHEMBL4456660)
Affinity DataIC50:  390nMAssay Description:Inhibition of APN on human ES-2 cell surface using L-Leu-p-nitroanilide as substrate after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed