BDBM50529326 CHEMBL4557197
SMILES Oc1cccn(CC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)OCc2ccccc2)c1=O
InChI Key InChIKey=PEFBFISDEVURKN-NRFANRHFSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50529326
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 5.70E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.85E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of human recombinant ERAP2 expressed in baculovirus infected Sf9 cells using omniMMP fluorogenic substrate incubated for 5 to 10 mins by f...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of human recombinant ERAP1 expressed in baculovirus infected Sf9 cells using omniMMP fluorogenic substrate incubated for 5 to 10 mins by f...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of human recombinant IRAP expressed in baculovirus infected Sf9 cells using omniMMP fluorogenic substrate incubated for 5 to 10 mins by fl...More data for this Ligand-Target Pair