BDBM50534731 CHEMBL4570214

SMILES CC1CCCCN1C\C=C\C(=O)N1CCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc12

InChI Key InChIKey=QOSRLQUTKKYXOX-QPJJXVBHSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50534731   

TargetEpidermal growth factor receptor(Homo sapiens (Human))
Jiangsu Aosaikang Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50534731(CHEMBL4570214)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of EGFR phosphorylation in EGF-stimulated human KB cells preincubated for 1 hr followed by EGF stimulation measured after 6 mins by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed