BDBM50536362 CHEMBL4517346
SMILES COc1ccccc1Nc1nc(cs1)-c1sc(NC(C)=O)nc1C
InChI Key InChIKey=ZADCDCMLLGDCRM-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50536362
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University Of Texas Southwestern Medical Center
Curated by ChEMBL
University Of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of MMP-9 (unknown origin) using Cys(Eu)-Pro-Leu-Gly-Leu-Lys(QSY7)-Ala-Arg-amide as substrate for 15 mins by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of human proMMP9 expressed in African green monkey COS-1 cells assessed as reduction in protein activation incubated for 30 mins prior to ...More data for this Ligand-Target Pair