BDBM50538840 CHEMBL4642925

SMILES CCOC(=O)c1cnc2ccc(nc2c1N[C@H]1CC[C@H](CO)CC1)-c1cc(Cl)c(O)c(Cl)c1

InChI Key InChIKey=ZBOWUNZOBLCBIG-CTYIDZIISA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50538840   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50538840(CHEMBL4642925)
Affinity DataEC50:  100nMAssay Description:Inhibition of human DYRK1A transfected in HEK293T cells co-transfected with Renilla plasmid, pGL3-NFAT and NFATc1 assessed as derepression of NFAT-de...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed