BDBM50558706 CHEMBL4750625
SMILES CCC(NC(=O)[C@H](Cc1ccc(O)c(c1)[N+]([O-])=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](N)CC(N)=O)C(N)=O
InChI Key InChIKey=LKQQKKQSOSJUFO-QOWIWEFOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50558706
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 6.72E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR1 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 2.84E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR5 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 6.07E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR3 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR4 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 3.75E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR2 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair