BDBM50560836 CHEMBL4758243

SMILES CCOC[C@H](COC(=O)CCc1ccccc1OCc1cccc(Oc2ccccc2)c1)OP(O)(=O)OC[C@H](N)C(O)=O

InChI Key InChIKey=PWIBLZZVGUIXAU-SXOMAYOGSA-N

Data  10 EC50

PDB links: 2 PDB IDs match this monomer.

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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50560836   

TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProbable G-protein coupled receptor 34(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Danio rerio)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50560836(CHEMBL4758243)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB