BDBM50566873 CHEMBL4859531

SMILES CN(C)Cc1ccc(CNC(=O)c2ccc3nncn3c2)cc1

InChI Key InChIKey=INYAZFZIPMYIQV-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50566873   

TargetProtein ENL(Homo sapiens)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566873(CHEMBL4859531)
Affinity DataIC50:  621nMAssay Description:Inhibition of human His-ENL YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetYEATS domain-containing protein 2(Homo sapiens)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566873(CHEMBL4859531)
Affinity DataIC50: >5.40E+4nMAssay Description:Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetYEATS domain-containing protein 4(Homo sapiens)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566873(CHEMBL4859531)
Affinity DataIC50: >5.40E+4nMAssay Description:Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566873(CHEMBL4859531)
Affinity DataIC50:  4.93E+3nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed