BDBM50571567 CHEMBL4847433
SMILES COc1ccc(CCc2nc3cc(ccn3c2NC(C)C)-c2c(C)noc2C)cc1OC
InChI Key InChIKey=RVEFPHKFXBBFEJ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50571567
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Massachusetts Boston
Curated by ChEMBL
University Of Massachusetts Boston
Curated by ChEMBL
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.51E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair