BDBM50582161 CHEMBL5076889
SMILES CC(=O)Nc1ccc(cc1)-n1nc2c(c1-c1oc3cc(ccc3c1C)C(=O)Nc1cccc(c1)C(F)(F)F)c(N)n[nH]c2=O
InChI Key InChIKey=GMVAILVBISMMBH-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50582161
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Bytedance Ai Lab
Curated by ChEMBL
Bytedance Ai Lab
Curated by ChEMBL
Affinity DataEC50: 34nMAssay Description:Inhibition of DDR1 in human THP-1 cells assessed as reduction in collagen induced DDR1 autophosphorylation by Western blot analysisMore data for this Ligand-Target Pair
TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Bytedance Ai Lab
Curated by ChEMBL
Bytedance Ai Lab
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human DDR1 (492 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by sc...More data for this Ligand-Target Pair