BDBM50586724 CHEMBL5082666
SMILES [O-][N+](=O)CC(c1c([nH]c2ccccc12)-c1ccsc1)c1ccccc1
InChI Key InChIKey=NCOQFHIDDWOEMQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50586724
Affinity DataKi: 43nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid scintillation spectrometry ana...More data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Positive allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as beta-arrestin 2 recruitment incubated for 90 mins by PathH...More data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Positive allosteric modulation of CB1 receptor in MF1 mouse vas deferens assessed as inhibition of AEA-induced electrically evoked vas deferens contr...More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cell membranes assessed as increase in [35S]GTPgammaS binding incubated for 30 mins by liquid...More data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:Positive allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP production incubated ...More data for this Ligand-Target Pair