BDBM50614127 CHEMBL5267043
SMILES CC(=O)N1c2cnc(NC(=O)OCC3(CC3)C(F)(F)F)nc2C2(CCC(F)(F)CC2)C1(C)C
InChI Key InChIKey=XEGSXAZIAWXAJO-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50614127
Affinity DataIC50: 48nMAssay Description:Antagonist activity at TSHR in rat FRTL-5 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 156nMAssay Description:Antagonist activity at human FSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human TSHR expressed in HEK293 cells assessed as reduction in cAMP production incubated for 2 hrs by Eu-cAMP tracer based TR-F...More data for this Ligand-Target Pair
Ligand Info