BDBM521420 6-(2-fluoro-4- methyl-phenyl)- 5-[2-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]oxypyrimidin- 5-yl]-8,9- dihydro-7H- benzo[7]annulen- 2-ol::US11149031, Example 244
SMILES Cc1ccc(c(F)c1)C1=C(c2cnc(O[C@H]3CCN(CCCF)C3)nc2)c2ccc(O)cc2CCC1
InChI Key InChIKey=HTQUXUFPCHDMRF-QHCPKHFHSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 521420
Affinity DataIC50: 3nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair