BDBM522079 US11155558, Compound 2g

SMILES CCCc1c(\C=N\O)n(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(CCO[N+]([O-])=O)CC1

InChI Key InChIKey=UWCJDXJUIYAAIP-WGOQTCKBSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 522079   

TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Topadur Pharma

US Patent
LigandPNGBDBM522079(US11155558, Compound 2g)
Affinity DataIC50:  1.00E+4nMAssay Description:The inhibition of recombinant human (rh) PDE5A by test compounds is measured in a radiometric assay based on Scintillation Proximity Assay (SPA) tech...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent