BDBM523803 US11136312, Compound SK-I-132
SMILES COc1cccc(Sc2nnc(Cc3c[nH]c4cc(F)ccc34)n2CCCc2c[nH]cn2)c1
InChI Key InChIKey=IBFJVEXBVBFLNC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 523803
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University
US Patent
Board of Trustees of The Southern Illinois University
US Patent
Affinity DataKi: 0.646nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University
US Patent
Board of Trustees of The Southern Illinois University
US Patent
Affinity DataKi: 656nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University
US Patent
Board of Trustees of The Southern Illinois University
US Patent
Affinity DataKi: 2.88E+3nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University
US Patent
Board of Trustees of The Southern Illinois University
US Patent
Affinity DataKi: 2.91E+3nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University
US Patent
Board of Trustees of The Southern Illinois University
US Patent
Affinity DataKi: >1.00E+4nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University
US Patent
Board of Trustees of The Southern Illinois University
US Patent
Affinity DataEC50: 0.992nMAssay Description:Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...More data for this Ligand-Target Pair