BDBM528565 2-((6-((5-chloro-2-((3S,5R)-3,5-dimethylpiperazin-1-yl)pyrimidin-4-yl)amino)-1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)oxy)-N-methylacetamide ::US11192880, Example X-1
SMILES CNC(=O)COc1cc2cc(Nc3nc(ncc3Cl)N3C[C@H](C)N[C@H](C)C3)ccc2n(C)c1=O
InChI Key InChIKey=NSSRTMPGNIDSTM-OKILXGFUSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 528565
TargetB-cell lymphoma 6 protein/B-cell lymphoma 6 protein [32-99]/Nuclear receptor corepressor 2(Homo sapiens (Human))
Ontario Institute For Cancer Research (Oicr)
US Patent
Ontario Institute For Cancer Research (Oicr)
US Patent
Affinity DataIC50: 1.60E+3nMAssay Description:This assay is used to determine whether compounds inhibit the interaction between the BTB domain of BCL6 and a peptide derived from the BCL6 binding ...More data for this Ligand-Target Pair