BDBM534097 6-(Azetidin-1-yl)-4-fluoro-N-(2,2,5,6-tetramethyl-2,3-dihydro-1-benzofuran-7-sulfonyl)-1-benzofuran-2-carboxamide::WO2022081807, Example 204

SMILES Cc1cc2CC(C)(C)Oc2c(c1C)S(=O)(=O)NC(=O)c1cc2c(F)cc(cc2o1)N1CCC1

InChI Key InChIKey=ZACOYCQNFGRNGO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 534097   

TargetHistone acetyltransferase KAT6A [507-778](Homo sapiens)
The Broad Institute

WIPO
LigandPNGBDBM534097(6-(Azetidin-1-yl)-4-fluoro-N-(2,2,5,6-tetramethyl-...)
Affinity DataIC50:  7.70nMAssay Description:Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-FR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed