BDBM540774 US11261211, Compound SA-90
SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](O)(CC[C@H]34)C(F)F)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2ccccc12
InChI Key InChIKey=IKDNMNYXNGZQKN-ATDMNIQZSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 540774
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Sage Therapeutics
US Patent
Sage Therapeutics
US Patent
Affinity DataIC50: 300nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair