BDBM546320 US11286268, Compound 2001

SMILES OC(=O)c1cccc(c1)-c1cc(Cl)ccc1OCCn1c(Nc2ccccc2)nc2c(Cl)nccc2c1=O

InChI Key InChIKey=XVJRZGRKVXYFPI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 546320   

TargetEukaryotic translation initiation factor 4E-binding protein 1(Human)
Effector Therapeutics

US Patent
LigandPNGBDBM546320(US11286268, Compound 2001)
Affinity DataIC50: 6.58E+4nMAssay Description:eIF4E protein was pre-incubated with EDA-m7GDP-ATTO-550 in FPB at 2xconcentrations for 5 minutes prior to the addition of compounds. Compounds (100x)...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2022
Entry Details
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