BDBM576088 N-(1-(4-chlorobenzyl)-2- methyl-6-(6-methyl-7-oxo-6,7- dihydro-1H-pyrrolo[2,3-c] pyridin-4-yl)-1H-benzo[d] imidazol-4-yl)ethane- sulfonamide::US11466034, Example 41
SMILES CCS(=O)(=O)Nc1cc(cc2n(Cc3ccc(Cl)cc3)c(C)nc12)-c1cn(C)c(=O)c2[nH]ccc12
InChI Key InChIKey=CDTQQFOUFQKDDX-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 576088
TargetBromodomain-containing protein 4 [349-460](Homo sapiens (Human))
Betta Pharmaceuticals
US Patent
Betta Pharmaceuticals
US Patent
Affinity DataIC50: 0.400nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair