BDBM618528 US20230287003, Example 5u
SMILES OC1CC2COCC(C1)N2c1ncc(Cl)c(Nc2ccc3n(CC4CC(F)(F)C4)c(=O)c4OCC[C@@H](Nc4c3c2)C2CC2)n1
InChI Key InChIKey=WJNBUCPPEQXGRP-KGQZTBJRSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 618528
Affinity DataIC50: 8.32nMAssay Description:Each 15 μL HTRF reaction in a 384-well black Proxiplate (Perkin Elmer) contained 1 nM Trx-6×His-BCL6 (in house-produced, human BCL6 BTB domain c...More data for this Ligand-Target Pair