BDBM618588 US20230287003, Example 13f
SMILES Cn1c2ccc(Nc3nc(ncc3Cl)N3CCN(CCC#N)CC3)cc2c2N[C@@H](C3CC3)C(F)(F)COc2c1=O
InChI Key InChIKey=OAUOEZLIBDIYKL-QHCPKHFHSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 618588
Affinity DataIC50: 2.19nMAssay Description:Each 15 μL HTRF reaction in a 384-well black Proxiplate (Perkin Elmer) contained 1 nM Trx-6×His-BCL6 (in house-produced, human BCL6 BTB domain c...More data for this Ligand-Target Pair