BDBM629782 US20230340011, Example 76.::US20230340011, Example 77.
SMILES C[C@H](CCC(=O)N1CCC[C@@H](C1)c1ccccc1)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C
InChI Key InChIKey=KDXIKDSGZQUKRE-VMJKVMBGSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 629782
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Asteroid Therapeutics
US Patent
Asteroid Therapeutics
US Patent
Affinity DataIC50: 125nMAssay Description:10,000 cells/well of the PathHunter U2OS SREBP-2 Nuclear Translocation Cell Line are plated in quadruplicate on 384 well plates in 20 μL of Assa...More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:PathHunter NHR CHO cells stably transfected with tagged full-length human LXRβ and a nuclear fusion protein containing Steroid Receptor Co-activ...More data for this Ligand-Target Pair
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Asteroid Therapeutics
US Patent
Asteroid Therapeutics
US Patent
Affinity DataIC50: 125nMAssay Description:10,000 cells/well of the PathHunter U2OS SREBP-2 Nuclear Translocation Cell Line are plated in quadruplicate on 384 well plates in 20 μL of Assa...More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:PathHunter NHR CHO cells stably transfected with tagged full-length human LXRβ and a nuclear fusion protein containing Steroid Receptor Co-activ...More data for this Ligand-Target Pair