BDBM71502 US9694002, 524

SMILES Fc1cc(CN2CCC(CC2)Oc2ncc(cc2Cl)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1

InChI Key InChIKey=LMRLMSNXUMMQMU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 71502   

TargetSodium channel protein type 1/10/11/2/3/4/5/8/9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM71502(US9694002, 524)
Affinity DataIC50:  11nMpH: 7.4 T: 2°CAssay Description:Binding of this radioligand was preformed in 5 mL borosilicate glass test tubes at room temperature. Binding was initiated by adding membranes to inc...More data for this Ligand-Target Pair
In DepthDetails US Patent