BDBM81510 JCP-666

SMILES OC(=O)CN(NC(=O)c1ccc(CNC(=O)c2cccc(c2)C(O)=O)cc1)C(=O)[C@H]1O[C@@H]1C(=O)N(Cc1cccc2ccccc12)Cc1cccc2ccccc12

InChI Key InChIKey=ASKNZQDJJSNTBW-YDAXCOIMSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 81510   

TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50:  1.38E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50: >7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50:  7.00E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed