BDBM81512 VEA-417

SMILES NC(=O)CNC(=O)c1ccc(cc1)C(=O)NNC(=O)[C@H]1O[C@@H]1C(=O)N(Cc1cccc2ccccc12)Cc1cccc2ccccc12

InChI Key InChIKey=FROMJEVAQJJCHT-ACHIHNKUSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 81512   

TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50:  3.25E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50: >7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50:  1.31E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed